hae_ʻaoʻao

huahana

Mea hana pauka Lemairamin (WGX-50) CAS No.: 29946-61-0 98.0% maʻemaʻe min. no nā mea hoʻohui

Wehewehe Pōkole:

He hui kūlohelohe ʻo Lemairamin a i ʻole Wgx50 i unuhi ʻia mai nā pepa chili i hōʻike i nā hopena maikaʻi i ka pale ʻana i ka maʻi Alzheimer. Ua ʻike ʻia nā haʻawina hiki iā ia ke kāohi i ka apoptosis neuronal i hoʻokomo ʻia e Aβ, hoʻēmi i ka ʻawahia calcium neuronal, a hoʻēmi i ka hōʻiliʻili ʻana o nā oligomers Aβ i loko o ka cerebral cortex.


Nā kikoʻī huahana

Nā Lepili Huahana

Wikiō Huahana

Nā Palena Huahana

Inoa huahana

ʻO Lemairamina

Inoa ʻē aʻe

2-Propenamide, N-[2-(3,4-dimethoxyphenyl)ethyl]-3-phenyl-, (2E)-;

ʻO Lemairamin (WGX-50)

Helu CAS.

29946-61-0

ʻO ke ʻano molekole

C19H21NO3

Kaumaha molekole

311.37

Maʻemaʻe

98.0%

helehelena

Pauka keʻokeʻo a keʻokeʻo paha

Noi

Mea Hoʻohui Meaʻai Maka

Hoʻolauna huahana

ʻO Lemairamin a i ʻole Wgx50 kahi hui kūlohelohe i unuhi ʻia mai nā pepa chili i hōʻike i nā hopena hoʻohiki i ka pale ʻana i ka maʻi Alzheimer. Ua ʻike ʻia nā haʻawina hiki iā ia ke kāohi i ka apoptosis neuronal i hoʻokomo ʻia e Aβ, hoʻēmi i ka ʻona calcium neuronal, a hoʻēmi i ka hōʻiliʻili ʻana o nā oligomers Aβ i loko o ka cortex cerebral. Eia kekahi, ua hōʻike ʻia ʻo wgx50 e hoʻomaikaʻi i ka hana cognitive i nā ʻiole. Hōʻike ka noiʻi he hiki iā wgx50 ke pale i ka hui ʻana o ka protein-protein ma waena o nā molekala amyloid. Ma keʻano holoʻokoʻa, loaʻa iā wgx50 ka hiki ke pale i ka maʻi Alzheimer a hiki ke hāʻawi i nā ala hou no ka hoʻomohala ʻana i nā lāʻau lapaʻau e kuhikuhi ana i nā oligomers Aβ. Eia kekahi, hōʻike ʻo WGX-50 i ka hana anti-inflammatory koʻikoʻi, ka mea e lilo ai ia i moho hoʻohiki no ka mālama ʻana i nā maʻi mumū. Ua ʻike ʻia he hopena koʻikoʻi ko WGX-50 i ka ʻili, e like me ka hoʻēmi ʻana i nā wrinkles a me ka hoʻomaikaʻi ʻana i ka elasticity o ka ʻili. Ma waho aʻe o nā hui kūlohelohe i unuhi ʻia mai ka mea kanu ʻo Zanthoxylum bungeanum, aia i kēia manawa nā hui synthetic i hoʻohana ʻia i nā noi like ʻole a ʻoi aku ka kūpono no ka mākeke.

Hiʻona

(1) Maʻemaʻe kiʻekiʻe: Hiki iā Lemairamin ke loaʻa nā huahana maʻemaʻe kiʻekiʻe ma o ka unuhi kūlohelohe a me nā kaʻina hana hoʻomaʻemaʻe. ʻO ke ʻano o ka maʻemaʻe kiʻekiʻe ʻo ia hoʻi ka bioavailability maikaʻi a me nā hopena ʻino liʻiliʻi.

(2) Palekana: Palekana kiʻekiʻe, kakaikahi nā hopena maikaʻi ʻole, ʻaʻohe hopena maikaʻi ʻole maopopo me ka hoʻohana lōʻihi.

(3) Paʻa: Loaʻa iā Lemairamin ke kūpaʻa maikaʻi a hiki ke mālama i kāna hana a me ka hopena ma lalo o nā ʻano like ʻole a me nā kūlana mālama.

(4) Maʻalahi ke omo: Hiki ke omo koke ʻia ʻo Lemairamin e ke kino o ke kanaka a hoʻolaha ʻia i nā ʻiʻo a me nā ʻōpū like ʻole.

Nā noi

ʻO Lemairamin kahi hui amide i unuhi ʻia mai ka ʻili o ka mea kanu Zanthoxylum bungeanum. Hoʻohana ʻia i kēia manawa ma ke ʻano he mea hoʻohui meaʻai, hana pū ia ma ke ʻano he agonist o ka alpha7 nicotinic acetylcholine receptor (α7nAChR), ka mea e hōʻemi ana i ka neuroinflammation i ka maʻi Alzheimer, a ua synthetic loa. Ua hōʻike ʻo Wgx50 i nā hopena hoʻoikaika i nā haʻawina preclinical, me ka pale ʻana i ka apoptosis neuronal i hoʻokomo ʻia e Aβ, ka hōʻemi ʻana i ka ʻona calcium neuronal, ka hōʻemi ʻana i ka hōʻiliʻili ʻana o nā oligomers Aβ i loko o ka cerebral cortex, a me ka hoʻomaikaʻi ʻana i ka hana cognitive i nā ʻiole.


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