Mea hana pauka hui 7P CAS No.: 1890208-58-8 99% maʻemaʻe min. no nā mea hoʻohui
Wikiō Huahana
Nā Palena Huahana
| Inoa huahana | Hui 7P |
| Inoa ʻē aʻe | Hui7P;2-[(2-methoxyphenyl)[(4-methylphenyl)sulfonyl]amino]-N-(4-methoxy-3-pyridinyl)acetamide; 2-(N-(2-methoxyphenyl)-4-methylphenylsulfonamido)-N-(4-methoxypyridin-3-yl)acetamide |
| Helu CAS. | 1890208-58-8 |
| ʻO ke ʻano molekole | C22H23N3O5S |
| Kaumaha molekole | 441.51 |
| Maʻemaʻe | 99.0% |
| helehelena | Pauka keʻokeʻo |
| Noi | Nootropic |
Hoʻolauna huahana
ʻO ka Hui 7P e pili ana i kahi hui organik kikoʻī e loaʻa ana i ʻehiku mau ʻātoma kalapona. I loko o ke kemika organik, he mea koʻikoʻi ke kalapona no ka mea hiki iā ia ke hana i nā pilina paʻa me nā ʻātoma ʻē aʻe, me nā ʻātoma kalapona, e hana i nā molekala paʻakikī. Hiki i kēia mau molekala ke loaʻa nā ʻano waiwai a me nā hana like ʻole, e hoʻolilo ana i nā hui i hoʻokumu ʻia i ke kalapona i mau poloka kūkulu o ke ola. I loko o nā hiʻohiʻona holoholona o ka ʻeha o ke aʻalolo optic, ua hōʻike ʻia ka hui 7p e hoʻoulu i ka ulu ʻana o nā axons GAP-43-positive, e hōʻike ana i ka hana ulu neurite o ka hui 7p in vitro e unuhi i ka hoʻoulu ʻana o ka hana hou axonal i vivo. ʻO ka pauka Hui 7P he pauka keʻokeʻo a keʻokeʻo paha i hana ʻia ma ke ʻano he hui tandem no ka ʻike ʻana i nā mea hoʻopaʻa antagonist thromboxane receptor dual-acting. ʻO ka ʻoiaʻiʻo, ua hōʻike ka hui 7p i ke koho ʻana no ka prostaglandin I2 synthase (PTGIS, CYP8A1) e pili ana i ka thromboxane synthase (CYP5A1). Hoʻolaha ka pauka hui nootropic 7P i ka ulu ʻana o nā axons Gap-43-positive, no laila e hoʻoulu ai i ka hana hou axonal i loko o ke kino. Ua hoʻolālā ʻia ka Complex 7p kiʻekiʻe e hoʻomaikaʻi i ka hoʻonohonoho ʻana, hoʻomaikaʻi i ke ʻano a kōkua i ka hakakā ʻana i ka luhi. Pale pū ia i ka oxidation o ka lolo a kōkua i ka hakakā ʻana i ka hōʻino ʻana o ka lolo i hoʻokumu ʻia e ka inu ʻana i ka waiʻona.
Hiʻona
(1) Maʻemaʻe kiʻekiʻe: Hiki i ka hui 7P ke loaʻa nā huahana maʻemaʻe kiʻekiʻe ma o nā kaʻina hana hana i hoʻomaʻemaʻe ʻia. ʻO ke ʻano o ka maʻemaʻe kiʻekiʻe ʻo ia hoʻi ka bioavailability maikaʻi a me nā hopena ʻino e emi ana.
(2) Palekana: Ua hōʻoia ʻia ka palekana o ka hui 7P no ke kino kanaka.
(3) Paʻa: Loaʻa i ka hui 7P ke kūpaʻa maikaʻi a hiki ke mālama i kāna hana a me ka hopena ma lalo o nā ʻano like ʻole a me nā kūlana mālama.
Nā noi
Hoʻonui ka Hui 7p i ka ulu ʻana o ka neurite o nā neurons mua i hoʻoulu ʻia mai ka hippocampus, cerebral cortex, a me ka retina a hoʻoulu i ka hana hou ʻana o nā aʻalolo optic i nā hiʻohiʻona holoholona o ka ʻeha o ke aʻalolo optic. Hoʻonui pū ia i ka hoʻonohonoho ʻana, mālama i ka hōʻino ʻana o ka lolo e pili ana i ka waiʻona, a pale i ka oxidation a puni ka lolo. Kōkua pū ia i ka hoʻomaikaʻi ʻana i ke ʻano a me ke kaua ʻana i ka luhi.












