Amino Tadalafil pauka mea hana CAS No.: 385769-84-6 98% maemae min.no nā mea hoʻohui
Nā Kūlana Huahana
Inoa mea kūʻai | Amino Tadalafil |
inoa ʻē aʻe | (6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3 ,4-b]indole-1,4(6H,7H)-dione |
CAS No. | 385769-84-6 |
ʻAno molekala | C21H18N4O4 |
Kaumaha molekula | 390.39 |
Maemae | 98.0% |
Ka nana aku | ʻO ka pauka keʻokeʻo keʻokeʻo |
Palapala noi | Mea ʻai meaʻai kumu |
Hoʻolauna huahana
ʻO Amino Tadalafil kahi hui like me Tadalafil, me kekahi o nā pūʻulu hana i loko o kona ʻano i hoʻololi ʻia e nā hui amino.ʻO ia ka PDE5 inhibitor a loaʻa nā hopena pharmacological e like me Tadalafil.Hoʻohana nui ia no ka mālama ʻana i ka male erectile dysfunction (ED).Ke hoʻohālikelike ʻia me Tadalafil, ʻoi aku ka lohi o ka metabolic rate o Amino Tadalafil i ke kino, a no laila hiki ke loaʻa ka hopena lōʻihi.
Hiʻona
(1) Ke koho kiʻekiʻe: Amino Tadalafil he kiʻekiʻe ke koho no PDE5, me kahi pilina kiʻekiʻe loa no PDE5 ma mua o nā subtypes PDE.ʻO kēia keʻano e hiki ai iā Amino Tadalafil ke pale aku i ka hana o ka enzyme PDE5, e hoʻoikaika i ke kahe o ke koko i loko o nā'ōpū hānau kāne a me ka hoʻomaikaʻiʻana i nā hōʻailona o ka erectile dysfunction (ED).
(2) Ka hopena lōʻihi: ʻO Amino Tadalafil ka wikiwiki o ka metabolism i loko o ke kino, e hiki ai iā ia ke hana i kahi hopena pharmacological lōʻihi loa, a hiki i nā hola 36.Hana kēia iā Amino Tadalafil i ka lāʻau lapaʻau ED lōʻihi, ʻaʻole pono e lawe pinepine ʻia.
(3) He liʻiliʻi nā hopena ʻaoʻao: ʻO Amino Tadalafil ka liʻiliʻi o nā hopena ʻaoʻao i hoʻohālikelike ʻia me Tadalafil, e like me ke poʻo ʻeha, a me ka ʻeha o ka ʻōpū.Ma muli o kāna koho kiʻekiʻe, hiki i ka Amino Tadalafil ke pale aku i nā pilina me nā subtypes PDE ʻē aʻe, e hōʻemi ana i ka hopena o nā hopena ʻaoʻao.
(4) Nā manaʻo hoʻohana ākea: Ma kahi o ka mālama ʻana iā ED, hiki ke hoʻohana ʻia ʻo Amino Tadalafil e mālama i nā maʻi ʻē aʻe e like me ka pulmonary arterial hypertension.ʻO kēia ka mea e loaʻa ai iā Amino Tadalafil nā noi noi ākea i ka wā e hiki mai ana.
Nā noi
ʻO Amino Tadalafil kahi hui i hoʻomohala ʻia i nā makahiki i hala iho nei, he ʻano like me Tadalafil, akā ua hoʻololi ʻia kekahi mau hui i loko o kāna ʻano e nā hui amino.I kēia manawa, ʻaʻole i ʻae ʻia ʻo Amino Tadalafil no ka hoʻohana ʻana i ka lāʻau lapaʻau, no laila ua palena iki kāna noi ʻana i ka lāʻau lapaʻau.Eia naʻe, ua hōʻike ʻia kekahi mau haʻawina e hiki ke hoʻohana ʻia kēia pūhui.
ʻO Amino Tadalafil he mea hoʻopiʻi PDE5, he hopena pharmacological like me Tadalafil.Hiki iā ia ke hoʻomaikaʻi i nā hōʻailona o ka erectile dysfunction (ED) ma o ka hoʻoikaika ʻana i ke kahe o ke koko i loko o nā ʻōpū hānau kāne ma ke kāohi ʻana i ka hana o ka enzyme PDE5.Ke hoʻohālikelikeʻia me Tadalafil,ʻo Amino Tadalafil ka wikiwiki o ka metabolism i loko o ke kino, hiki ke loaʻa ka hopena mau loa.ʻO kēia ka mea i loaʻa iā Amino Tadalafil ka mana nui i ka mālama ʻana iā ED.
Eia kekahi, hiki ke hoʻohana ʻia ʻo Amino Tadalafil e mālama i kekahi mau maʻi ʻē aʻe, e like me ka hypertension arterial pulmonary.Ua hōʻike kekahi mau haʻawina e hiki i nā mea hoʻopaneʻe PDE5 ke hoʻonui i nā kīʻaha koko pulmonary, ma laila e hoʻomaikaʻi ai i nā hōʻailona o nā maʻi me ka hypertension arterial pulmonary.No ka mea he hopena pharmacological like ʻo Amino Tadalafil e like me Tadalafil, hiki ke hoʻohana ʻia e mālama i ka hypertension arterial pulmonary.
Ma keʻano holoʻokoʻa, loaʻa iā Amino Tadalafil ka mana hoʻohana nui, akā pono nā hoʻokolohua lapaʻau hou e hoʻoholo ai i kona palekana a me ka pono.Inā hāʻawi kēia mau ho'āʻo i nā hopena maikaʻi, hiki ke lilo ʻo Amino Tadalafil i lāʻau lapaʻau hou no ka mālama ʻana i ka ED a me ka hypertension arterial pulmonary, e hāʻawi ana i nā koho lapaʻau hou aku no nā kauka lapaʻau a me nā maʻi.