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Amino Tadalafil pauka mea hana CAS No.: 385769-84-6 98% maemae min.no nā mea hoʻohui

ʻO ka wehewehe pōkole:

ʻO Amino Tadalafil kahi hui like me Tadalafil, me kekahi o nā pūʻulu hana i loko o kona ʻano i hoʻololi ʻia e nā hui amino.


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Amino Tadalafil

inoa ʻē aʻe

(6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[ 3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A -Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dione;(6R,12aR)-2-Amino-6-(benzo[d][1,3] ]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R ,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3 ,4-b]indole-1,4(6H,7H)-dione

CAS No.

385769-84-6

ʻAno molekala

C21H18N4O4

Kaumaha molekula

390.39

Maemae

98.0%

Ka nana aku

ʻO ka pauka keʻokeʻo keʻokeʻo

Palapala noi

Mea ʻai meaʻai kumu

Hoʻolauna huahana

ʻO Amino Tadalafil kahi hui like me Tadalafil, me kekahi o nā pūʻulu hana i loko o kona ʻano i hoʻololi ʻia e nā hui amino.ʻO ia ka PDE5 inhibitor a loaʻa nā hopena pharmacological e like me Tadalafil.Hoʻohana nui ia no ka mālama ʻana i ka male erectile dysfunction (ED).Ke hoʻohālikelike ʻia me Tadalafil, ʻoi aku ka lohi o ka metabolic rate o Amino Tadalafil i ke kino, a no laila hiki ke loaʻa ka hopena lōʻihi.

Hiʻona

(1) Ke koho kiʻekiʻe: Amino Tadalafil he kiʻekiʻe ke koho no PDE5, me kahi pilina kiʻekiʻe loa no PDE5 ma mua o nā subtypes PDE.ʻO kēia keʻano e hiki ai iā Amino Tadalafil ke pale aku i ka hana o ka enzyme PDE5, e hoʻoikaika i ke kahe o ke koko i loko o nā'ōpū hānau kāne a me ka hoʻomaikaʻiʻana i nā hōʻailona o ka erectile dysfunction (ED).

(2) Ka hopena lōʻihi: ʻO Amino Tadalafil ka wikiwiki o ka metabolism i loko o ke kino, e hiki ai iā ia ke hana i kahi hopena pharmacological lōʻihi loa, a hiki i nā hola 36.Hana kēia iā Amino Tadalafil i ka lāʻau lapaʻau ED lōʻihi, ʻaʻole pono e lawe pinepine ʻia.

(3) He liʻiliʻi nā hopena ʻaoʻao: ʻO Amino Tadalafil ka liʻiliʻi o nā hopena ʻaoʻao i hoʻohālikelike ʻia me Tadalafil, e like me ke poʻo ʻeha, a me ka ʻeha o ka ʻōpū.Ma muli o kāna koho kiʻekiʻe, hiki i ka Amino Tadalafil ke pale aku i nā pilina me nā subtypes PDE ʻē aʻe, e hōʻemi ana i ka hopena o nā hopena ʻaoʻao.

(4) Nā manaʻo hoʻohana ākea: Ma kahi o ka mālama ʻana iā ED, hiki ke hoʻohana ʻia ʻo Amino Tadalafil e mālama i nā maʻi ʻē aʻe e like me ka pulmonary arterial hypertension.ʻO kēia ka mea e loaʻa ai iā Amino Tadalafil nā noi noi ākea i ka wā e hiki mai ana.

Nā noi

ʻO Amino Tadalafil kahi hui i hoʻomohala ʻia i nā makahiki i hala iho nei, he ʻano like me Tadalafil, akā ua hoʻololi ʻia kekahi mau hui i loko o kāna ʻano e nā hui amino.I kēia manawa, ʻaʻole i ʻae ʻia ʻo Amino Tadalafil no ka hoʻohana ʻana i ka lāʻau lapaʻau, no laila ua palena iki kāna noi ʻana i ka lāʻau lapaʻau.Eia naʻe, ua hōʻike ʻia kekahi mau haʻawina e hiki ke hoʻohana ʻia kēia pūhui.

ʻO Amino Tadalafil he mea hoʻopiʻi PDE5, he hopena pharmacological like me Tadalafil.Hiki iā ia ke hoʻomaikaʻi i nā hōʻailona o ka erectile dysfunction (ED) ma o ka hoʻoikaika ʻana i ke kahe o ke koko i loko o nā ʻōpū hānau kāne ma ke kāohi ʻana i ka hana o ka enzyme PDE5.Ke hoʻohālikelikeʻia me Tadalafil,ʻo Amino Tadalafil ka wikiwiki o ka metabolism i loko o ke kino, hiki ke loaʻa ka hopena mau loa.ʻO kēia ka mea i loaʻa iā Amino Tadalafil ka mana nui i ka mālama ʻana iā ED.

Eia kekahi, hiki ke hoʻohana ʻia ʻo Amino Tadalafil e mālama i kekahi mau maʻi ʻē aʻe, e like me ka hypertension arterial pulmonary.Ua hōʻike kekahi mau haʻawina e hiki i nā mea hoʻopaneʻe PDE5 ke hoʻonui i nā kīʻaha koko pulmonary, ma laila e hoʻomaikaʻi ai i nā hōʻailona o nā maʻi me ka hypertension arterial pulmonary.No ka mea he hopena pharmacological like ʻo Amino Tadalafil e like me Tadalafil, hiki ke hoʻohana ʻia e mālama i ka hypertension arterial pulmonary.

Ma keʻano holoʻokoʻa, loaʻa iā Amino Tadalafil ka mana hoʻohana nui, akā pono nā hoʻokolohua lapaʻau hou e hoʻoholo ai i kona palekana a me ka pono.Inā hāʻawi kēia mau ho'āʻo i nā hopena maikaʻi, hiki ke lilo ʻo Amino Tadalafil i lāʻau lapaʻau hou no ka mālama ʻana i ka ED a me ka hypertension arterial pulmonary, e hāʻawi ana i nā koho lapaʻau hou aku no nā kauka lapaʻau a me nā maʻi.


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