Mea hana pauka Galantamine Hydrobromide CAS No.: 1953-04-4 98% maʻemaʻe min. no nā mea hoʻohui
Nā Palena Huahana
| Inoa huahana | ʻO Galantamine Hydrobromide |
| Inoa ʻē aʻe | ʻO Galanthamine hydrobromide; ʻO Galantamine HBr; Galanthamine HBr;(4aS,6R,8aS) -4a,5,9,10,11,12-hexahydro-3-methoxy-11-methyl-6H-Benzofuro[3a,3,2-ef][2]benzazepin-6-ol, Hydrobromide |
| Helu CAS. | 1953-04-4 |
| ʻO ke ʻano molekole | C17H21NO3.HBr |
| Kaumaha molekole | 368.27 |
| Maʻemaʻe | 98.0% |
| helehelena | pauka keʻokeʻo a keʻokeʻo paha |
| Hoʻopili ʻana | 1kg/ʻeke 10kgs, 25kgs/pahu |
| Noi | nā lāʻau nootropic |
Hoʻolauna huahana
ʻO Galantamine hydrobromide kahi benzazepine i loaʻa mai nā ʻōpuʻu a me nā pua o narcissus, osmanthus, a i ʻole canna. He mea hoʻopale cholinesterase waha nō hoʻi ia. Ma ke ʻano he ligand no nā mea loaʻa acetylcholine nicotinic, ua hoʻohana nui ʻia ia e hoʻoikaika i ka hana neurocognitive. ʻO kāna hana ka hoʻokūkū a me ka hoʻohuli ʻana i ka acetylcholinesterase, a laila e hoʻonui ai i ka nui o ka acetylcholine. Ke komo i loko o ke koko, ua komo koke ka galantamine hydrobromide i nā ʻāpana like ʻole o ke kino, me ka lolo. Hoʻopaʻa ia i nā mea loaʻa acetylcholine nicotinic, e hoʻololi ana i ke ʻano a hoʻonui i ka hoʻokuʻu ʻana o acetylcholine. Hana pū ia ma ka hoʻokūkū ʻana a me ka hoʻohuli ʻana i nā hopena o nā mea hoʻopale cholinesterase. Ma ka pale ʻana i ka cholinesterase, pale ia i ka haki ʻana o ka acetylcholine, a laila e hoʻonui ai i nā pae a me ka lōʻihi o kēia neurotransmitter ikaika. Hiki iā Galantamine ke hoʻomaikaʻi i ke aʻo ʻana a me ka hoʻomanaʻo, pale i ka mumū o ka lolo, a mālama i nā pae kiʻekiʻe o nā neurotransmitters ma ka mālama ʻana i ka pono o nā neurons a me nā synapses.
Hiʻona
(1) Maʻemaʻe kiʻekiʻe: Hiki i ka Galantamine hydrobromide ke lilo i huahana maʻemaʻe kiʻekiʻe ma o nā kaʻina hana hoʻomaʻemaʻe. ʻO ke ʻano o ka maʻemaʻe kiʻekiʻe ʻo ia hoʻi ka bioavailability maikaʻi a me nā hopena ʻino liʻiliʻi.
(2) Palekana: Ua hōʻoia ʻia ʻo Galantamine hydrobromide he palekana no ke kino kanaka.
(3) Paʻa: Loaʻa i ka Galantamine hydrobromide ke kūpaʻa maikaʻi a hiki ke mālama i kāna hana a me ka hopena ma lalo o nā ʻano like ʻole a me nā kūlana mālama.
Nā noi
Ma ke ʻano he mea hoʻohui meaʻai, hiki i ka galantamine hydrobromide ke hoʻomaikaʻi i ka hoʻomanaʻo, ka ʻike, a me ka hiki ke hana i nā hana o kēlā me kēia lā. Hana ia ma ka hoʻihoʻi ʻana i ke kaulike o kekahi mau mea kūlohelohe (neurotransmitters) i loko o ka lolo, kahi e hoʻonui ai i ka wikiwiki o ka hoʻokumu ʻana i ka hoʻomanaʻo a hoʻomaikaʻi i ka paʻa ʻana o nā kikoʻī a me nā ʻoiaʻiʻo. Eia kekahi, hoʻopilikia pololei a ʻaʻole pololei paha ka galantamine hydrobromide i ka neuroplasticity. Hoʻoulu ia i ka plasticity synaptic ma ka hoʻoulu ʻana i nā microglia a me nā astrocytes. Hāʻawi ʻo Galantamine i ka pale antioxidant e kūʻē i ke kaumaha oxidative i hoʻokumu ʻia e nā radical free.












